List of sulfonamides

Short description: None

This is a list of sulfonamides used in medicine.

## Contents

* 1 Antimicrobials
* 2 Sulfonylureas (anti-diabetic agents)
* 3 Diuretics
* 4 Anticonvulsants
* 5 Dermatologicals
* 6 Antiretrovirals
* 7 Hepatitis C antivirals
* 8 Stimulants
* 9 NSAIDs
* 10 Cardiac and Vasoactive Medications
* 11 Triptans
* 12 Others
* 13 References
* 14 External links

## Antimicrobials

Short-acting[1]

* Sulfacetamide
* Sulfadiazine
* Sulfadimidine
* Sulfafurazole (sulfisoxazole)
* Sulfisomidine (sulfaisodimidine)
* Sulfaguanidine

Intermediate-acting

* Sulfamethoxazole[2]
* Sulfamoxole
* Sulfanitran

Long-acting

* Sulfadimethoxine
* Sulfamethoxypyridazine
* Sulfametoxydiazine

Ultra long-acting

* Sulfadoxine
* Sulfametopyrazine
* Terephtyl

## Sulfonylureas (anti-diabetic agents)

* Acetohexamide
* Carbutamide
* Chlorpropamide
* Glibenclamide (glyburide)
* Glibornuride
* Gliclazide
* Glyclopyramide
* Glimepiride
* Glipizide
* Gliquidone
* Glisoxepide
* Glicaramide
* Tolazamide
* Tolbutamide

## Diuretics

* Acetazolamide
* Bumetanide
* Chlorthalidone
* Chlorothiazide
* Clopamide
* Furosemide
* Hydrochlorothiazide
* Indapamide
* Mefruside
* Metolazone
* Xipamide
* Methazolamide
* Torasemide

## Anticonvulsants

* Ethoxzolamide
* Sultiame
* Zonisamide

## Dermatologicals

* Mafenide

## Antiretrovirals

* Amprenavir (HIV protease inhibitor)
* Darunavir (HIV protease inhibitor)
* Delavirdine (non-nucleoside reverse transcriptase inhibitor)
* Fosamprenavir (HIV protease inhibitor)
* Tipranavir (HIV protease inhibitor)

## Hepatitis C antivirals

* Asunaprevir (NS3/4A protease inhibitor)
* Beclabuvir (NS5B RNA polymerase inhibitor)
* Dasabuvir (NS5B RNA polymerase inhibitor)
* Grazoprevir (NS3/4A protease inhibitor)
* Paritaprevir (NS3/4A protease inhibitor)
* Simeprevir (NS3/4A protease inhibitor)

## Stimulants

* Azabon

## NSAIDs

* Apricoxib (COX-2 inhibitor)
* Celecoxib (COX-2 inhibitor)
* Parecoxib (COX-2 inhibitor)

## Cardiac and Vasoactive Medications

* Bosentan (endothelin receptor antagonist)
* Diazoxide (insulin release inhibitor and vasodilator)
* Dofetilide (class III antiarrhythmic)
* Dronedarone (class III antiarrhythmic)
* Ibutilide (class III antiarrhythmic)
* Sotalol (β blocker)
* Tamsulosin (α blocker)
* Udenafil (PDE5 inhibitor)

## Triptans

* Almotriptan (antimigraine)
* Sumatriptan (antimigraine)
* Naratriptan (antimigraine)

## Others

* Brinzolamide (carbonic anhydrase inhibitor for glaucoma)
* Dorzolamide (anti-glaucoma carbonic anhydrase inhibitor)
* Famotidine (histamine H2 receptor antagonist)
* Probenecid (uricosuric)
* Sulfasalazine (anti-inflammatory agent and a DMARD)
* Vemurafenib (anticancer B-Raf inhibitor)

## References

1. ↑ Brayfield, A, ed (2 February 2011). "Sulfonamides and diaminopyrimidines". Martindale: The Complete Drug Reference. Pharmaceutical Press. http://www.medicinescomplete.com/mc/martindale/current/1-a16-10-g.htm. Retrieved 28 March 2014.
2. ↑ Tripathi, K. D. (2019). Essentials of medical pharmacology (Eighth ed.). New Delhi: Jaypee Brothers Medical Publishers. ISBN 978-93-5270-499-6.

## External links

* ~~List of sulfonamides~~
* Author of The Demon Under the Microscope, a history of the discovery of the sulfa drugs
* A History of the Fight Against Tuberculosis in Canada (Chemotherapy)
* Presentation speech, Nobel Prize in Physiology and Medicine, 1939
* The History of WW II Medicine
* "Five Medical Miracles of the Sulfa Drugs". Popular Science, June 1942, pp. 73–78.
* A history of antibiotics

* v
* t
* e

Antibacterials: nucleic acid inhibitors (J01E, J01M)

Antifolates
(inhibits
purine metabolism,
thereby inhibiting
DNA and RNA synthesis)|

| DHFR inhibitor|

* 2,4-Diaminopyrimidine
* Trimethoprim#
* Brodimoprim
* Tetroxoprim
* Iclaprim†

|

Sulfonamides
(DHPS inhibitor)|

| Short-
acting|

* Sulfaisodimidine
* Sulfamethizole
* Sulfadimidine
* Sulfapyridine
* Sulfafurazole
* Sulfanilamide
* Prontosil
* Sulfathiazole
* Sulfathiourea

|

Intermediate-
acting|

* Sulfamethoxazole
* Sulfadiazine#
* Sulfamoxole

Long-
acting|

* Sulfadimethoxine
* Sulfadoxine
* Sulfalene
* Sulfametomidine
* Sulfametoxydiazine
* Sulfamethoxypyridazine
* Sulfaperin
* Sulfamerazine
* Sulfaphenazole
* Sulfamazone

Other/ungrouped|

* Sulfacetamide
* Sulfadicramide
* Sulfametrole
* Sulfanitran

Combinations|

* Trimethoprim/sulfamethoxazole#
* Ormetoprim/sulfadimethoxine

Other DHPS inhibitors|

* Dapsone

Topoisomerase
inhibitors/
quinolones/
(inhibits
DNA replication)|

| 1st g.|

* Cinoxacin‡
* Flumequine‡
* Nalidixic acid‡
* Oxolinic acid‡
* Pipemidic acid‡
* Piromidic acid‡
* Rosoxacin‡

|

Fluoro-
quinolones|

| 2nd g.|

* Ciprofloxacin#
* Ofloxacin
* Enoxacin‡
* Fleroxacin‡
* Lomefloxacin‡
* Nadifloxacin‡
* Norfloxacin‡
* Pefloxacin‡
* Rufloxacin‡

|

3rd g.|

* Levofloxacin#
* Balofloxacin‡
* Grepafloxacin‡
* Pazufloxacin‡
* Sparfloxacin‡
* Temafloxacin‡
* Tosufloxacin‡

4th g.|

* Besifloxacin
* Delafloxacin
* Gatifloxacin
* Finafloxacin
* Gemifloxacin
* Moxifloxacin#
* Clinafloxacin†
* Garenoxacin‡
* Prulifloxacin‡
* Sitafloxacin‡
* Trovafloxacin‡/Alatrofloxacin‡

Vet.|

* Danofloxacin
* Difloxacin
* Enrofloxacin
* Ibafloxacin
* Marbofloxacin
* Orbifloxacin
* Pradofloxacin
* Sarafloxacin‡

Newer non-fluorinated|

* Nemonoxacin

Related (DG)|

* Aminocoumarins: Novobiocin

Anaerobic DNA
inhibitors|

| Nitro- imidazole derivatives|

* Metronidazole#
* Tinidazole
* Ornidazole

|

Nitrofuran derivatives|

* Nitrofurantoin#
* Furazolidone‡
* Nifurtoinol

RNA synthesis|

| Rifamycins/
RNA polymerase|

* Rifampicin#
* Rifabutin#
* Rifapentine#
* Rifaximin
* Rifalazil§

|

Lipiarmycins|

* Fidaxomicin

* #WHO-EM
* ‡Withdrawn from market
* Clinical trials:
* †Phase III
* §Never to phase III

* v
* t
* e

Anticonvulsants (N03)

GABAergics|

| GABAAR PAMs|

* Barbiturates: Barbexaclone
* Metharbital
* Methylphenobarbital
* Pentobarbital
* Phenobarbital#
* Primidone; Carbamates: Felbamate; Benzodiazepines: Clobazam
* Clonazepam
* Clorazepate
* Diazepam#
* Lorazepam#
* Midazolam
* Nimetazepam
* Nitrazepam
* Temazepam; Others: Bromide (potassium bromide, sodium bromide)
* Imepitoin
* Paraldehyde
* Stiripentol

|

GABA-T inhibitors|

* Fatty acids (and related): Valproate
* Valpromide
* Valproate pivoxil
* Vigabatrin

Others|

* GABAR agonists: Progabide; GAT-1 inhibitors: Tiagabine

Channel
modulators|

| Sodium blockers|

* Hydantoins: Ethotoin
* Fosphenytoin
* Mephenytoin
* Phenytoin#; Ureides: Acetylpheneturide
* Chlorphenacemide
* Phenacemide‡
* Pheneturide; Fatty acids: Valproate
* Valpromide
* Valproate pivoxil; Carboxamides: Carbamazepine#
* Eslicarbazepine acetate
* Oxcarbazepine; Others: Lacosamide
* Lamotrigine#
* Rufinamide
* Topiramate
* Zonisamide

|

Calcium blockers|

* Oxazolidinediones: Ethadione
* Paramethadione
* Trimethadione; Succinimides: Ethosuximide#
* Mesuximide
* Phensuximide; Gabapentinoids: Gabapentin
* Pregabalin; Others: Imepitoin
* Lamotrigine#
* Topiramate
* Zonisamide

Potassium openers|

* Retigabine

Others|

| CA inhibitors|

* Sulfonamides: Acetazolamide
* Ethoxzolamide
* Sultiame
* Topiramate
* Zonisamide

|

Others|

* Albutoin
* Beclamide
* Brivaracetam
* Cannabidiol
* Etiracetam
* Levetiracetam
* Perampanel

* #WHO-EM
* ‡Withdrawn from market
* Clinical trials:
* †Phase III
* §Never to phase III

* v
* t
* e

Antibiotics and chemotherapeutics for dermatological use (D06)

Antibiotics|

| Tetracycline and derivatives|

* Demeclocycline
* Chlortetracycline
* Oxytetracycline
* Tetracycline

|

Others|

* Amphenicol: Chloramphenicol

* Aminoglycosides: Neomycin
* Gentamicin
* Amikacin

* Quinolones: Nadifloxacin

* Streptogramin: Virginiamycin

* Rifamycin: Rifaximin

* other: Fusidic acid
* Bacitracin
* Tyrothricin
* Mupirocin

Chemotherapeutics|

| Sulfonamides|

* Silver sulfadiazine
* Sulfathiazole
* Mafenide
* Sulfamethizole
* Sulfanilamide
* Sulfamerazine

|

Antivirals|

* Aciclovir
* Penciclovir
* Idoxuridine
* Edoxudine
* Imiquimod
* Resiquimod
* Podophyllotoxin
* Docosanol
* Tromantadine
* Inosine
* Lysozyme
* Ibacitabine
* Lysine

Other|

* Ingenol mebutate
* Metronidazole

* v
* t
* e

Antihypertensives: diuretics (C03)

Sulfonamides
(and etacrynic acid)|

| CA inhibitors (at PT)|

* Acetazolamide

|

Loop (Na-K-Cl at AL)|

* Furosemide#
* Azosemide
* Bumetanide
* Etacrynic acid
* Etozolin
* Muzolimine
* Ozolinone
* Piretanide
* Tienilic acid
* Torasemide

[[Chemistry:ThiThiazides (Sodium-chloride Na-Cl at Distal convoluted tubule|DCT]],
Calcium-sparing)|

* Altizide
* Bendroflumethiazide
* Butizide
* Chlorothiazide
* Cyclopenthiazide
* Cyclothiazide
* Epitizide
* Hydrochlorothiazide#
* Hydroflumethiazide
* Mebutizide
* Methyclothiazide
* Polythiazide
* Trichlormethiazide

Thiazide-likes (primarily DCT)|

* Quinethazone
* Clopamide
* Chlortalidone
* Mefruside
* Clofenamide
* Metolazone
* Meticrane
* Xipamide
* Indapamide
* Clorexolone
* Fenquizone

Potassium-sparing (at CD)|

| ESC blockers|

* Amiloride#
* Triamterene
* Benzamil

|

Aldosterone antagonists|

* Spirolactones
* Spironolactone#
* Eplerenone
* Potassium canrenoate
* Canrenone

* Nonsteroidal
* Finerenone

Osmotic diuretics (PT, DL)|

* Mannitol#
* Glycerol
* Urea

Vasopressin receptor inhibitors
(DCT and CD)|

* Vaptans
* Conivaptan
* Mozavaptan
* Satavaptan
* Tolvaptan

* Others
* Demeclocycline
* Lithium carbonate

Other|

* Ethanol, Isopropanol, 2M2B
* mercurial diuretics (Chlormerodrin, Mersalyl, Meralluride)
* Theobromine
* Cicletanine

* #WHO-EM
* ‡Withdrawn from market
* Clinical trials:
* †Phase III
* §Never to phase III

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