Testosterone Nicotinate

Testosterone nicotinate
Clinical data
Trade names	Bolfortan, Linobol
Other names	WD-53
Routes of; administration	Intramuscular injection
Identifiers
	IUPAC name (1S,2R,10R,11S,14S,15S)-2,15-dimethyl-5-oxotetracyclo[8.7.0.02,7.011,15]heptadec-6-en-14-yl pyridine-3-carboxylate;
CAS Number	668-56-4;
PubChem CID	101826;
ChemSpider	91999;
UNII	44F122YR9Q;
Chemical and physical data
Formula	C25H31NO3
Molar mass	393.527 g·mol−1
3D model (JSmol)	Interactive image;
	SMILES C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2OC(=O)C4=CN=CC=C4)CCC5=CC(=O)CC[C@]35C;
	InChI InChI=1S/C25H31NO3/c1-24-11-9-18(27)14-17(24)5-6-19-20-7-8-22(25(20,2)12-10-21(19)24)29-23(28)16-4-3-13-26-15-16/h3-4,13-15,19-22H,5-12H2,1-2H3/t19-,20-,21-,22-,24-,25-/m0/s1; Key:KHRRLLSDLVLEIT-BKWLFHPQSA-N;

Short description: Chemical compound

Testosterone nicotinate (brand names Bolfortan, Linobol) is an androgen and anabolic steroid medication made by esterifying nicotinic acid and testosterone^[1]^[2]^[3]^[4]^[5] It was formulated as a 50 mg/mL aqueous suspension provided in ampoules.^[4]^[5] The medication was manufactured and sold by Lannacher Heilmittel GmbH in Austria.^[5] It is no longer marketed.^[5]

Testosterone nicotinate had a relatively short duration, somewhere between that of testosterone propionate and testosterone enanthate.^[5]^[4]

References

↑ The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. 14 November 2014. pp. 641–642. ISBN 978-1-4757-2085-3. https://books.google.com/books?id=0vXTBwAAQBAJ&pg=PA641.
↑ Index Nominum 2000: International Drug Directory. Taylor & Francis. January 2000. ISBN 978-3-88763-075-1. https://books.google.com/books?id=5GpcTQD_L2oC&pg=PA976.
↑ Concise Dictionary of Pharmacological Agents: Properties and Synonyms. Springer Science & Business Media. 6 December 2012. ISBN 978-94-011-4439-1. https://books.google.com/books?id=tsjrCAAAQBAJ&pg=PA270.
↑ ^4.0 ^4.1 ^4.2 Virginia. Task Force on Anabolic Steroid Misuse Among Minors (1988). Report of the Task Force on Anabolic Steroid Misuse Among Minors: To the Director, Virginia Department of Health Regulatory Boards. Department of Health Regulatory Boards. https://books.google.com/books?id=KGHZAAAAMAAJ. "BOLFORTAN injection 50mgs/cc 1 ampules Lanniker Heilmittel, Austria cc Bolfortan is an nicotinate. The nicotinate added to the steroid molecule makes it last longer than regular [...] make this short, aqueous testosterone testosterone aqueous, although being water based, this form of testosterone gets into the system rather quickly. Testosterone Nicotinate has a half-life somewhere between Testosterone Propionate and Testosterone Enanthate."
↑ ^5.0 ^5.1 ^5.2 ^5.3 ^5.4 Anabolics. Molecular Nutrition LLC. 2011. pp. 182–184. ISBN 978-0-9828280-1-4. https://books.google.com/books?id=afKLA-6wW0oC&pg=PP182.

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(incl. AAS)

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  | group1 = AR antagonists
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| list2 =

  | group3 = Antigonadotropins
  | list3 =

D₂ receptor antagonists (prolactin releasers) (e.g., domperidone, metoclopramide, risperidone, haloperidol, chlorpromazine, sulpiride)
Estrogens (e.g., bifluranol, [[diethylstilbestrol, estradiol, estradiol esters, ethinylestradiol, ethinylestradiol sulfonate, paroxypropione)
GnRH agonists (e.g., leuprorelin)
GnRH antagonists (e.g., cetrorelix)
Progestogens (incl., chlormadinone acetate, [[cyproterone acetate, hydroxyprogesterone caproate, gestonorone caproate, [[Chemistry:Medroxyprogesterone medroxyprogesterone acetate, Chemistry:Megestrol acetate|megestrol acetate]])

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Androstenedione immunogens: Androvax (androstenedione albumin)
Ovandrotone albumin (Fecundin)

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^#WHO-EM
^‡Withdrawn from market
Clinical trials:
- ^†Phase III
- ^§Never to phase III

See also: Androgen receptor modulators; Estrogens and antiestrogens; Progestogens and antiprogestogens; List of androgens/anabolic steroids

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Original source: https://en.wikipedia.org/wiki/Testosterone nicotinate. Read more

[Elks2014-1] The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. 14 November 2014. pp. 641–642. ISBN 978-1-4757-2085-3. https://books.google.com/books?id=0vXTBwAAQBAJ&pg=PA641.

[IndexNominum2000-2] Index Nominum 2000: International Drug Directory. Taylor & Francis. January 2000. ISBN 978-3-88763-075-1. https://books.google.com/books?id=5GpcTQD_L2oC&pg=PA976.

[MortonHall2012-3] Concise Dictionary of Pharmacological Agents: Properties and Synonyms. Springer Science & Business Media. 6 December 2012. ISBN 978-94-011-4439-1. https://books.google.com/books?id=tsjrCAAAQBAJ&pg=PA270.

[Minors1988-4] 4.0 ^4.1 ^4.2 Virginia. Task Force on Anabolic Steroid Misuse Among Minors (1988). Report of the Task Force on Anabolic Steroid Misuse Among Minors: To the Director, Virginia Department of Health Regulatory Boards. Department of Health Regulatory Boards. https://books.google.com/books?id=KGHZAAAAMAAJ. "BOLFORTAN injection 50mgs/cc 1 ampules Lanniker Heilmittel, Austria cc Bolfortan is an nicotinate. The nicotinate added to the steroid molecule makes it last longer than regular [...] make this short, aqueous testosterone testosterone aqueous, although being water based, this form of testosterone gets into the system rather quickly. Testosterone Nicotinate has a half-life somewhere between Testosterone Propionate and Testosterone Enanthate."

[Llewellyn2011-5] 5.0 ^5.1 ^5.2 ^5.3 ^5.4 Anabolics. Molecular Nutrition LLC. 2011. pp. 182–184. ISBN 978-0-9828280-1-4. https://books.google.com/books?id=afKLA-6wW0oC&pg=PP182.

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5α-Reductase	Alfatradiol Dutasteride Epristeride Finasteride Saw palmetto extract
Others	Abiraterone acetate Aminoglutethimide Bifluranol Cyproterone acetate Flutamide Ketoconazole Nilutamide Seviteronel^† Spironolactone

Testosterone Nicotinate

See also

References