List Of Sulfonamides

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This is a list of sulfonamides used in medicine.

Antimicrobials

Short-acting^[1]

Intermediate-acting

Long-acting

Ultra long-acting

Sulfadoxine
Sulfametopyrazine
Terephtyl

Sulfonylureas (anti-diabetic agents)

Diuretics

Anticonvulsants

Dermatologicals

Mafenide

Antiretrovirals

Amprenavir (HIV protease inhibitor)
Darunavir (HIV protease inhibitor)
Delavirdine (non-nucleoside reverse transcriptase inhibitor)
Fosamprenavir (HIV protease inhibitor)
Tipranavir (HIV protease inhibitor)

Hepatitis C antivirals

Asunaprevir (NS3/4A protease inhibitor)
Beclabuvir (NS5B RNA polymerase inhibitor)
Dasabuvir (NS5B RNA polymerase inhibitor)
Grazoprevir (NS3/4A protease inhibitor)
Paritaprevir (NS3/4A protease inhibitor)
Simeprevir (NS3/4A protease inhibitor)

Stimulants

Azabon

NSAIDs

Apricoxib (COX-2 inhibitor)
Celecoxib (COX-2 inhibitor)
Parecoxib (COX-2 inhibitor)

Cardiac and Vasoactive Medications

Bosentan (endothelin receptor antagonist)
Diazoxide (insulin release inhibitor and vasodilator)
Dofetilide (class III antiarrhythmic)
Dronedarone (class III antiarrhythmic)
Ibutilide (class III antiarrhythmic)
Sotalol (β blocker)
Tamsulosin (α blocker)
Udenafil (PDE5 inhibitor)

Triptans

Almotriptan (antimigraine)
Sumatriptan (antimigraine)
Naratriptan (antimigraine)

Others

Brinzolamide (carbonic anhydrase inhibitor for glaucoma)
Dorzolamide (anti-glaucoma carbonic anhydrase inhibitor)
Famotidine (histamine H₂ receptor antagonist)
Probenecid (uricosuric)
Sulfasalazine (anti-inflammatory agent and a DMARD)
Vemurafenib (anticancer B-Raf inhibitor)

References

↑ Brayfield, A, ed (2 February 2011). "Sulfonamides and diaminopyrimidines". Martindale: The Complete Drug Reference. Pharmaceutical Press. http://www.medicinescomplete.com/mc/martindale/current/1-a16-10-g.htm. Retrieved 28 March 2014.
↑ Tripathi, K. D. (2019). Essentials of medical pharmacology (Eighth ed.). New Delhi: Jaypee Brothers Medical Publishers. ISBN 978-93-5270-499-6.

External links

~~List of sulfonamides~~
Author of The Demon Under the Microscope, a history of the discovery of the sulfa drugs
A History of the Fight Against Tuberculosis in Canada (Chemotherapy)
Presentation speech, Nobel Prize in Physiology and Medicine, 1939
The History of WW II Medicine
"Five Medical Miracles of the Sulfa Drugs". Popular Science, June 1942, pp. 73–78.
A history of antibiotics

Antibacterials: nucleic acid inhibitors (J01E, J01M)

Antifolates
(inhibits
purine metabolism,
thereby inhibiting
DNA and RNA synthesis)

2,4-Diaminopyrimidine
- Trimethoprim^#
- Brodimoprim
- Tetroxoprim
- Iclaprim^†

Sulfonamides
(DHPS inhibitor)

Short- acting	Sulfaisodimidine Sulfamethizole Sulfadimidine Sulfapyridine Sulfafurazole Sulfanilamide Prontosil Sulfathiazole Sulfathiourea
Intermediate- acting	Sulfamethoxazole Sulfadiazine^# Sulfamoxole
Long- acting	Sulfadimethoxine Sulfadoxine Sulfalene Sulfametomidine Sulfametoxydiazine Sulfamethoxypyridazine Sulfaperin Sulfamerazine Sulfaphenazole Sulfamazone
Other/ungrouped	Sulfacetamide Sulfadicramide Sulfametrole Sulfanitran

Combinations

Other DHPS inhibitors

Dapsone

Topoisomerase
inhibitors/
quinolones/
(inhibits
DNA replication)

Fluoro-
quinolones

2nd g.	Ciprofloxacin^# Ofloxacin Enoxacin^‡ Fleroxacin^‡ Lomefloxacin^‡ Nadifloxacin^‡ Norfloxacin^‡ Pefloxacin^‡ Rufloxacin^‡
3rd g.	Levofloxacin^# Balofloxacin^‡ Grepafloxacin^‡ Pazufloxacin^‡ Sparfloxacin^‡ Temafloxacin^‡ Tosufloxacin^‡
4th g.	Besifloxacin Delafloxacin Gatifloxacin Finafloxacin Gemifloxacin Moxifloxacin^# Clinafloxacin^† Garenoxacin^‡ Prulifloxacin^‡ Sitafloxacin^‡ Trovafloxacin^‡/Alatrofloxacin^‡
Vet.	Danofloxacin Difloxacin Enrofloxacin Ibafloxacin Marbofloxacin Orbifloxacin Pradofloxacin Sarafloxacin^‡

Newer non-fluorinated

Nemonoxacin

Related (DG)

Aminocoumarins: Novobiocin

Anaerobic DNA
inhibitors

Nitro- imidazole derivatives	Metronidazole^# Tinidazole Ornidazole
Nitrofuran derivatives	Nitrofurantoin^# Furazolidone^‡ Nifurtoinol

RNA synthesis

Rifamycins/ RNA polymerase	Rifampicin^# Rifabutin^# Rifapentine^# Rifaximin Rifalazil^§
Lipiarmycins	Fidaxomicin

^#WHO-EM
^‡Withdrawn from market
Clinical trials:
- ^†Phase III
- ^§Never to phase III

Anticonvulsants (N03)

GABA_AR PAMs	Barbiturates: Barbexaclone Metharbital Methylphenobarbital Pentobarbital Phenobarbital^# Primidone; Carbamates: Felbamate; Benzodiazepines: Clobazam Clonazepam Clorazepate Diazepam^# Lorazepam^# Midazolam Nimetazepam Nitrazepam Temazepam; Others: Bromide (potassium bromide, sodium bromide) Imepitoin Paraldehyde Stiripentol
GABA-T inhibitors	Fatty acids (and related): Valproate Valpromide Valproate pivoxil Vigabatrin
Others	GABAR agonists: Progabide; GAT-1 inhibitors: Tiagabine

Channel
modulators

Sodium blockers	Hydantoins: Ethotoin Fosphenytoin Mephenytoin Phenytoin^#; Ureides: Acetylpheneturide Chlorphenacemide Phenacemide^‡ Pheneturide; Fatty acids: Valproate Valpromide Valproate pivoxil; Carboxamides: Carbamazepine^# Eslicarbazepine acetate Oxcarbazepine; Others: Lacosamide Lamotrigine^# Rufinamide Topiramate Zonisamide
Calcium blockers	Oxazolidinediones: Ethadione Paramethadione Trimethadione; Succinimides: Ethosuximide^# Mesuximide Phensuximide; Gabapentinoids: Gabapentin Pregabalin; Others: Imepitoin Lamotrigine^# Topiramate Zonisamide
Potassium openers	Retigabine

Others

CA inhibitors	Sulfonamides: Acetazolamide Ethoxzolamide Sultiame Topiramate Zonisamide
Others	Albutoin Beclamide Brivaracetam Cannabidiol Etiracetam Levetiracetam Perampanel

^#WHO-EM
^‡Withdrawn from market
Clinical trials:
- ^†Phase III
- ^§Never to phase III

Antibiotics and chemotherapeutics for dermatological use (D06)

Tetracycline and derivatives	Demeclocycline Chlortetracycline Oxytetracycline Tetracycline
Others	Amphenicol: Chloramphenicol Aminoglycosides: Neomycin Gentamicin Amikacin Quinolones: Nadifloxacin Streptogramin: Virginiamycin Rifamycin: Rifaximin other: Fusidic acid Bacitracin Tyrothricin Mupirocin

Chemotherapeutics

Sulfonamides	Silver sulfadiazine Sulfathiazole Mafenide Sulfamethizole Sulfanilamide Sulfamerazine
Antivirals	Aciclovir Penciclovir Idoxuridine Edoxudine Imiquimod Resiquimod Podophyllotoxin Docosanol Tromantadine Inosine Lysozyme Ibacitabine Lysine
Other	Ingenol mebutate Metronidazole

Antihypertensives: diuretics (C03)

Sulfonamides
(and etacrynic acid)

CA inhibitors (at PT)	Acetazolamide
Loop (Na-K-Cl at AL)	Furosemide^# Azosemide Bumetanide Etacrynic acid Etozolin Muzolimine Ozolinone Piretanide Tienilic acid Torasemide
[[Chemistry:ThiThiazides (Sodium-chloride Na-Cl at Distal convoluted tubule\|DCT]], Calcium-sparing)	Altizide Bendroflumethiazide Butizide Chlorothiazide Cyclopenthiazide Cyclothiazide Epitizide Hydrochlorothiazide^# Hydroflumethiazide Mebutizide Methyclothiazide Polythiazide Trichlormethiazide
Thiazide-likes (primarily DCT)	Quinethazone Clopamide Chlortalidone Mefruside Clofenamide Metolazone Meticrane Xipamide Indapamide Clorexolone Fenquizone

Potassium-sparing (at CD)

ESC blockers	Amiloride^# Triamterene Benzamil
Aldosterone antagonists	Spirolactones Spironolactone^# Eplerenone Potassium canrenoate Canrenone Nonsteroidal Finerenone

Osmotic diuretics (PT, DL)

Vasopressin receptor inhibitors
(DCT and CD)

Vaptans

Others
- Demeclocycline
- Lithium carbonate

Other

Ethanol, Isopropanol, 2M2B
mercurial diuretics (Chlormerodrin, Mersalyl, Meralluride)
Theobromine
Cicletanine

^#WHO-EM
^‡Withdrawn from market
Clinical trials:
- ^†Phase III
- ^§Never to phase III

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Categories: [Disulfiram-like drugs] [Hepatotoxins] [Sulfonamide antibiotics]

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